{"id":107188,"date":"2011-04-03T00:00:00","date_gmt":"2011-04-03T00:00:00","guid":{"rendered":"https:\/\/www.deberes.net\/tesis\/sin-categoria\/nuevas-dianas-en-esquizofrenia-diseno-y-sa%c2%adntese-de-nuevos-ligandos-selectivos-del-receptor-d3-de-dopamina\/"},"modified":"2011-04-03T00:00:00","modified_gmt":"2011-04-03T00:00:00","slug":"nuevas-dianas-en-esquizofrenia-diseno-y-sa%c2%adntese-de-nuevos-ligandos-selectivos-del-receptor-d3-de-dopamina","status":"publish","type":"post","link":"https:\/\/www.deberes.net\/tesis\/santiago-de-compostela\/nuevas-dianas-en-esquizofrenia-diseno-y-sa%c2%adntese-de-nuevos-ligandos-selectivos-del-receptor-d3-de-dopamina\/","title":{"rendered":"Nuevas dianas en esquizofrenia. dise\u00f1o y s\u00edntese de nuevos ligandos selectivos del receptor d3 de dopamina"},"content":{"rendered":"<h2>Tesis doctoral de <strong> Raquel Ortega Mart\u00ednez <\/strong><\/h2>\n<p>Debido a su localizaci\u00f3n y farmacolog\u00eda, los receptores dopamin\u00e9rgicos d3 pueden desempe\u00f1ar un papel en la fisiopatolog\u00eda de enfermedades del snc tales como la esquizofrenia y pueden representar una nueva diana de f\u00e1rmacos para el tratamiento de esta enfermedad. Diversos antagonistas selectivos d3 han mostrados eficacia en varios modelos predictivos de actividad antipsic\u00f3tica sin inducci\u00f3n de catalepsia o incremento de los niveles de prolactina plasm\u00e1tica. Un antagonista selectivo d3 podr\u00eda as\u00ed disminuir tanto los s\u00edntomas positivos como los negativos de la enfermedad, y no producir\u00eda los efectos secundarios asociados a las actuales terapias est\u00e1ndar (ej. Olanzapina). El objetivo de este proyecto es el desarrollo de nuevos ligandos (agonistas parciales y antagonistas) selectivos del receptor d3 que nos permitan establecer la importancia de este receptor en patolog\u00edas como la esquizofrenia.<\/p>\n<p>&nbsp;<\/p>\n<h3>Datos acad\u00e9micos de la tesis doctoral \u00ab<strong>Nuevas dianas en esquizofrenia. dise\u00f1o y s\u00edntese de nuevos ligandos selectivos del receptor d3 de dopamina<\/strong>\u00ab<\/h3>\n<ul>\n<li><strong>T\u00edtulo de la tesis:<\/strong>\u00a0 Nuevas dianas en esquizofrenia. dise\u00f1o y s\u00edntese de nuevos ligandos selectivos del receptor d3 de dopamina <\/li>\n<li><strong>Autor:<\/strong>\u00a0 Raquel Ortega Mart\u00ednez <\/li>\n<li><strong>Universidad:<\/strong>\u00a0 Santiago de compostela<\/li>\n<li><strong>Fecha de lectura de la tesis:<\/strong>\u00a0 04\/03\/2011<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n<h3>Direcci\u00f3n y tribunal<\/h3>\n<ul>\n<li><strong>Director de la tesis<\/strong>\n<ul>\n<li>Jorge  Christian Fern\u00e1ndez Masaguer<\/li>\n<\/ul>\n<\/li>\n<li><strong>Tribunal<\/strong>\n<ul>\n<li>Presidente del tribunal: Antonio Espinosa \u00fabeda <\/li>\n<li>hugo Gutierrez de teran casta\u00f1on (vocal)<\/li>\n<li>M\u00aa de los \u00e1ngeles Mart\u00edn hern\u00e1ndez (vocal)<\/li>\n<li>Elena Fern\u00e1ndez guti\u00e9rrez (vocal)<\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Tesis doctoral de Raquel Ortega Mart\u00ednez Debido a su localizaci\u00f3n y farmacolog\u00eda, los receptores dopamin\u00e9rgicos d3 pueden desempe\u00f1ar un papel [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center 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