{"id":11873,"date":"2001-02-07T00:00:00","date_gmt":"2001-02-07T00:00:00","guid":{"rendered":"https:\/\/www.deberes.net\/tesis\/sin-categoria\/analisis-de-la-interaccion-risperidona-neurotransmisores-en-diversas-preparaciones-de-musculo-liso\/"},"modified":"2001-02-07T00:00:00","modified_gmt":"2001-02-07T00:00:00","slug":"analisis-de-la-interaccion-risperidona-neurotransmisores-en-diversas-preparaciones-de-musculo-liso","status":"publish","type":"post","link":"https:\/\/www.deberes.net\/tesis\/ciencias-medicas\/analisis-de-la-interaccion-risperidona-neurotransmisores-en-diversas-preparaciones-de-musculo-liso\/","title":{"rendered":"An\u00e1lisis de la interacci\u00f3n risperidona-neurotransmisores en diversas preparaciones de musculo liso"},"content":{"rendered":"<h2>Tesis doctoral de <strong>  Nieto Bayon F\u00e9lix Manuel <\/strong><\/h2>\n<p>La risperidona es un f\u00e1rmaco neurol\u00e9ptico at\u00edpico que tiene una zona manejable m\u00e1s amplia que la de los antipsic\u00f3tiocs tric\u00edclicos y no tric\u00edclicos cl\u00e1sicos, produce m\u00ednimos efectos de tipo anticolin\u00e9rgico y no provoca apenas efectos cardiovascualres ni alteraciones de la conducci\u00f3n cardiaca.  material y m\u00e9todos  se utlizaron preparaciones de conducto deferente aislado de rata para el estudio de las interacciones de la risperidona con noradrenalian y dopamina; \u00fatero aislado de rata para el estudio de las interacciones con histamina, serotonina y oxitocina e ileon aislado de cobaya para las interacciones de risperidona con acetilcolina, 4-aminopiridina, potasio e histamina. se determi\u00f3 el valor de la concentraci\u00f3n inhibitoria 50 (ci50) y el valor de pd2 cuando el antagonismoera de tipo no competitivo.  resultados y discusi\u00f3n  la risperidona antagoniza de forma no competitiva las respuestas del conducto deferente aislado de rata a noradrenalina y dopamina cuando el medio de incubaci\u00f3n es soluci\u00f3n de krebs-henseleit normal; cuando a este medio de incubaci\u00f3n se a\u00f1ade: coca\u00edna, 17 beta estradiol y propranolol contin\u00faa manifest\u00e1ndose el antagonismo no competitivo existente entre la risperidona y la noradrenalina y la dopamina. La risperidona a las concentracion es ensayadas antagoniza de forma no competitiva los efectos de histamina, 4-aminopiridina y potasio en la preparaci\u00f3n de ileon aislado de cobaya. la risperidona a las concentraciones ensayadas antagoniza de forma no competitiva la respuesta del \u00fatero aislado de rata a serotonina e histamina, pero no a oxitocina y al ion potasio.  estos experimentos sugieren que la risperidona a concentraciones elevadas se comporta como f\u00e1rmaco estabilizador inespec\u00edfico de membrana, a pesar de no presentar isosterimos con los neurol\u00e9pticos ni con los antidepresivos tric\u00edclicos conocidos estabilizadores de membrana.<\/p>\n<p>&nbsp;<\/p>\n<h3>Datos acad\u00e9micos de la tesis doctoral \u00ab<strong>An\u00e1lisis de la interacci\u00f3n risperidona-neurotransmisores en diversas preparaciones de musculo liso<\/strong>\u00ab<\/h3>\n<ul>\n<li><strong>T\u00edtulo de la tesis:<\/strong>\u00a0 An\u00e1lisis de la interacci\u00f3n risperidona-neurotransmisores en diversas preparaciones de musculo liso <\/li>\n<li><strong>Autor:<\/strong>\u00a0  Nieto Bayon F\u00e9lix Manuel <\/li>\n<li><strong>Universidad:<\/strong>\u00a0 Valladolid<\/li>\n<li><strong>Fecha de lectura de la tesis:<\/strong>\u00a0 02\/07\/2001<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n<h3>Direcci\u00f3n y tribunal<\/h3>\n<ul>\n<li><strong>Director de la tesis<\/strong>\n<ul>\n<li>Alfonso Velasco Martin<\/li>\n<\/ul>\n<\/li>\n<li><strong>Tribunal<\/strong>\n<ul>\n<li>Presidente del tribunal: pedro S\u00e1nchez Garc\u00eda <\/li>\n<li>angela Alsasua del valle (vocal)<\/li>\n<li>cecilio \u00e1lamo gonz\u00e1lez (vocal)<\/li>\n<li>Luis San rom\u00e1n del barrio (vocal)<\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Tesis doctoral de Nieto Bayon F\u00e9lix Manuel La risperidona es un f\u00e1rmaco neurol\u00e9ptico at\u00edpico que tiene una zona manejable m\u00e1s [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center 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