{"id":132135,"date":"1996-01-01T00:00:00","date_gmt":"1996-01-01T00:00:00","guid":{"rendered":"https:\/\/www.deberes.net\/tesis\/sin-categoria\/estudio-farmacologico-de-nuevos-antagonistas-de-receptores-de-colecistoquinina\/"},"modified":"1996-01-01T00:00:00","modified_gmt":"1996-01-01T00:00:00","slug":"estudio-farmacologico-de-nuevos-antagonistas-de-receptores-de-colecistoquinina","status":"publish","type":"post","link":"https:\/\/www.deberes.net\/tesis\/ciencias-medicas\/estudio-farmacologico-de-nuevos-antagonistas-de-receptores-de-colecistoquinina\/","title":{"rendered":"Estudio farmacologico de nuevos antagonistas de receptores de colecistoquinina."},"content":{"rendered":"<h2>Tesis doctoral de <strong>  Ballaz Garcia Santiago Jes\u00fas <\/strong><\/h2>\n<p>La colecistoquinina (cck) es un peptido gastrointestinal y un neurotransmisor del sistema nervioso central. La utilizacion de antagonistas de cck es de gran interes terapeutico en el tratamiento de patolog\u00edas del aparato digestivo y en transtornos de ansiedad. En el presente trabajo se han desarrollado una nueva serie de antagonistas de naturaleza piridopirimidinica con gran afinidad y selectividad por los receptores de cck del tipo cck-a. Estos compuestos inhiben efectos fisiologicos mediados por la cck en preparaciones \u00abin vitro\u00bb como es la estimulacion de amilasa en suspensiones de acinos pancreaticos y la contraccion de preparaciones de plexo mienterico-musculo liso de ileon. En estudios \u00abin vivo\u00bb revierten tanto la hipofagia como la hipomotilidad inducidas por la administracion periferica de cck. Por ultimo el compuesto e-3, el mas potente de los estudiados, presenta una potente accion ansiolitica en los tests de vogel y de la caja de dos compartimentos de valoracion de ansiedad.<\/p>\n<p>&nbsp;<\/p>\n<h3>Datos acad\u00e9micos de la tesis doctoral \u00ab<strong>Estudio farmacologico de nuevos antagonistas de receptores de colecistoquinina.<\/strong>\u00ab<\/h3>\n<ul>\n<li><strong>T\u00edtulo de la tesis:<\/strong>\u00a0 Estudio farmacologico de nuevos antagonistas de receptores de colecistoquinina. <\/li>\n<li><strong>Autor:<\/strong>\u00a0  Ballaz Garcia Santiago Jes\u00fas <\/li>\n<li><strong>Universidad:<\/strong>\u00a0 Navarra<\/li>\n<li><strong>Fecha de lectura de la tesis:<\/strong>\u00a0 01\/01\/1996<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n<h3>Direcci\u00f3n y tribunal<\/h3>\n<ul>\n<li><strong>Director de la tesis<\/strong>\n<ul>\n<li>Ana Barber C\u00e1rcamo<\/li>\n<\/ul>\n<\/li>\n<li><strong>Tribunal<\/strong>\n<ul>\n<li>Presidente del tribunal: Francisco Ponz Piedrafita <\/li>\n<li>Gin\u00e9s Salido Ruiz (vocal)<\/li>\n<li>Edurne Cenarruzabeitia Sagarminaga (vocal)<\/li>\n<li> Garcia Lopez Mar\u00eda  Teresa (vocal)<\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Tesis doctoral de Ballaz Garcia Santiago Jes\u00fas La colecistoquinina (cck) es un peptido gastrointestinal y un neurotransmisor del sistema nervioso [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center 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