{"id":136434,"date":"2026-01-12T16:56:50","date_gmt":"2026-01-12T16:56:50","guid":{"rendered":"https:\/\/www.deberes.net\/tesis\/sin-categoria\/mecanismos-especializados-de-transporte-y-sus-interacciones-baclofeno\/"},"modified":"2026-01-12T16:56:50","modified_gmt":"2026-01-12T16:56:50","slug":"mecanismos-especializados-de-transporte-y-sus-interacciones-baclofeno","status":"publish","type":"post","link":"https:\/\/www.deberes.net\/tesis\/ciencias-medicas\/mecanismos-especializados-de-transporte-y-sus-interacciones-baclofeno\/","title":{"rendered":"Mecanismos especializados de transporte y sus interacciones: baclofeno."},"content":{"rendered":"<h2>Tesis doctoral de <strong> Ana Polache Vengut <\/strong><\/h2>\n<p>Con el fin de esclarecer la naturaleza de los portadores involucrados en el proceso de absorcion del baclofeno, se han realizado ensayos de inhibicion cruzados con el farmaco, y un compuesto relacionado estructuralmente: la beta-alanina. Los resultados obtenidos muestran que la beta-alanina se absorbe en intestino delgado de rata segun una cinetica saturable de michaelis-menten y que, efectivamente, actua como inhibidor competitivo de la absorcion del baclofeno.  teniendo en cuenta que los beta-aminoacidos no son componentes habituales de la dieta, no es de esperar que la presencia de alimentos en lumen intestinal conduzca a una reduccion significativa de la absorcion del baclofeno. No obstante, los peptidos peque\u00f1os presentes en intestino, podrian generar por hidrolisis beta-aminoacidos que tambien interferirian en la absorcion del farmaco. Por ello, seria conveniente prescribir el baclofeno entre comidas, particularmente en aquellos casos en que su administracion es critica, como ocurre en la esclerosis multiple.<\/p>\n<p>&nbsp;<\/p>\n<h3>Datos acad\u00e9micos de la tesis doctoral \u00ab<strong>Mecanismos especializados de transporte y sus interacciones: baclofeno.<\/strong>\u00ab<\/h3>\n<ul>\n<li><strong>T\u00edtulo de la tesis:<\/strong>\u00a0 Mecanismos especializados de transporte y sus interacciones: baclofeno. <\/li>\n<li><strong>Autor:<\/strong>\u00a0 Ana Polache Vengut <\/li>\n<li><strong>Universidad:<\/strong>\u00a0 Universitat de val\u00e9ncia (estudi general)<\/li>\n<li><strong>Fecha de lectura de la tesis:<\/strong>\u00a0 01\/01\/1991<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n<h3>Direcci\u00f3n y tribunal<\/h3>\n<ul>\n<li><strong>Director de la tesis<\/strong>\n<ul>\n<li> Pla Delfina  Jos\u00e9 M<\/li>\n<\/ul>\n<\/li>\n<li><strong>Tribunal<\/strong>\n<ul>\n<li>Presidente del tribunal: Victor Jimenez Torres <\/li>\n<li>Jos\u00e9 Bruno Fari\u00f1a Espinosa (vocal)<\/li>\n<li>Joaqu\u00edn Timoneda Timoneda (vocal)<\/li>\n<li>Daniel Fos Galve (vocal)<\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Tesis doctoral de Ana Polache Vengut Con el fin de esclarecer la naturaleza de los portadores involucrados en el proceso [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center 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