{"id":79751,"date":"2006-03-05T00:00:00","date_gmt":"2006-03-05T00:00:00","guid":{"rendered":"https:\/\/www.deberes.net\/tesis\/sin-categoria\/analisis-y-aplicacion-de-estrategias-para-el-descubrimiento-de-farmacos-sa%c2%adntesis-qsar-y-modelizacion-basada-en-el-receptor\/"},"modified":"2006-03-05T00:00:00","modified_gmt":"2006-03-05T00:00:00","slug":"analisis-y-aplicacion-de-estrategias-para-el-descubrimiento-de-farmacos-sa%c2%adntesis-qsar-y-modelizacion-basada-en-el-receptor","status":"publish","type":"post","link":"https:\/\/www.deberes.net\/tesis\/quimica-organica\/analisis-y-aplicacion-de-estrategias-para-el-descubrimiento-de-farmacos-sa%c2%adntesis-qsar-y-modelizacion-basada-en-el-receptor\/","title":{"rendered":"An\u00e1lisis y aplicaci\u00f3n de estrategias para el descubrimiento de f\u00e1rmacos: s\u00edntesis, qsar y modelizaci\u00f3n basada en el receptor"},"content":{"rendered":"<h2>Tesis doctoral de <strong> Santiago Vilar Varela <\/strong><\/h2>\n<p>En la presente tesis doctoral se han desarrollado modelos te\u00f3ricos de predicci\u00f3n de la actividad anti-vih y vasodilatadora mediante la utilizaci\u00f3n de m\u00e9todos de c\u00e1lculo de descriptores moleculares en combinaci\u00f3n con t\u00e9cnicas estad\u00edsticas para establecer una relaci\u00f3n entre la estructura molecular y la actividad biol\u00f3gica (m\u00e9todos qsar). Tambi\u00e9n se han realizado c\u00e1lculos de interacci\u00f3n f\u00e1rmaco-receptor mediante metodolog\u00edas de tipo docking y se ha realizado una s\u00edntesis org\u00e1nica de una serie de cumarinas an\u00e1logas al resveratol con una buena actividad vasodilatadora.<\/p>\n<p>&nbsp;<\/p>\n<h3>Datos acad\u00e9micos de la tesis doctoral \u00ab<strong>An\u00e1lisis y aplicaci\u00f3n de estrategias para el descubrimiento de f\u00e1rmacos: s\u00edntesis, qsar y modelizaci\u00f3n basada en el receptor<\/strong>\u00ab<\/h3>\n<ul>\n<li><strong>T\u00edtulo de la tesis:<\/strong>\u00a0 An\u00e1lisis y aplicaci\u00f3n de estrategias para el descubrimiento de f\u00e1rmacos: s\u00edntesis, qsar y modelizaci\u00f3n basada en el receptor <\/li>\n<li><strong>Autor:<\/strong>\u00a0 Santiago Vilar Varela <\/li>\n<li><strong>Universidad:<\/strong>\u00a0 Santiago de compostela<\/li>\n<li><strong>Fecha de lectura de la tesis:<\/strong>\u00a0 03\/05\/2006<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n<h3>Direcci\u00f3n y tribunal<\/h3>\n<ul>\n<li><strong>Director de la tesis<\/strong>\n<ul>\n<li>Eugenio Uriarte Villares<\/li>\n<\/ul>\n<\/li>\n<li><strong>Tribunal<\/strong>\n<ul>\n<li>Presidente del tribunal: bernardo Celda mu\u00f1oz <\/li>\n<li>humberto Gonz\u00e1lez d\u00edez (vocal)<\/li>\n<li>ram\u00f3n Garc\u00eda domenech (vocal)<\/li>\n<li>stefano Moro (vocal)<\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Tesis doctoral de Santiago Vilar Varela En la presente tesis doctoral se han desarrollado modelos te\u00f3ricos de predicci\u00f3n de la [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center 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